Full-text resources of PSJD and other databases are now available in the new Library of Science.
Visit https://bibliotekanauki.pl

PL EN


Preferences help
enabled [disable] Abstract
Number of results
2020 | 30 | 2 | 213-219

Article title

Design and Antimicrobial evaluation of 1-(2-(2,3,5-triphenylcyclopenta-2,4-dien-1-yl)ethyl)piperazine and their derivatives

Content

Title variants

Languages of publication

EN

Abstracts

EN
A total of six of 1,2,4,5-tetrasubstituted imidazoles were prepared by multicomponent cyclo- condensation of benzil, aromatic aldehyde, aminoethylpiperazine and ammonium acetate. The prepared compounds were screened for their antibacterial activity against S. aureus, S. typhi, E.coli and Pseudomonas and antifungal activity against A. niger, C. albicans, Rhizopus sp, and Mucor. They exhibited better activities against all the tested bacterial and fungal strains.

Year

Volume

30

Issue

2

Pages

213-219

Physical description

Contributors

  • Department of Chemistry, St. Joseph University, Nagaland - 797 115, India
author
  • Department of Chemistry, Thiruvalluvar University College of Arts and Science, Kallakurichi - 606213, India
  • Department of Chemistry, CK College of Engineering and Technology, Cuddalore - 607003, India
  • Department of Chemistry, Annamalai University, Annamalainagar - 608 002, India
author
  • Department of Chemistry, Pavai Arts and Science College for Women, Namkkal - 637401, Tamil Nadu, India

References

  • [1] L. Seifert, M. Harbeck, A. Thomas, N. Hoke, L. Zoller, I. Wiechmann, G. Grupe, H. C. Scholz and J. M. Riehm. PLoS One, 2013, 8, e75742
  • [2] O. Ruuskanen, E. Lahti, L. C. Jennings and D. R. Murdoch. Lancet, 2011, 377, 1264
  • [3] WHO Tuberculosis Factsheet, World Health Organization, March 2010.
  • [4] H. W. Boucher, G. H. Talbot, J. S. Bradley, J. E. Edwards, D. Gilbert, L. B. Rice, M. Scheld, B. Spellberg and J. Bartlett. Clin. Infect. Dis. 2009, 48, 1
  • [5] R.J. Scheffler, S. Colmer, H. Tyman, A.L. Demain and V.P. Gullo. Appl. Microbiol. Biotechnol. 2013, 97, 969
  • [6] L. Zhang, X.M. Peng, G.L.V. Damu, R.X. Geng and C.H. Zhou, Med. Res. Rev. 2014, 34, 340.
  • [7] X.M. Peng, G.L.V. Damu and C.H. Zhou. Curr. Pharm. Des. 2013, 19, 3884-3930
  • [8] H. Z. Zhang, Z. L. Zhao and C. H. Zhou, Eur. J. Med. Chem. 2018, 144, 444
  • [9] J. Akhtar, A. A. Khan, Z. Ali, R. Haider and M. S. Yar. Eur. J. Med. Chem. 2017, 125, 143
  • [10] Y. Hu, Y. F. Shen, X. H. Wu, X. Tu and G. X. Wang. Eur. J. Med. Chem, 2018, 143 958.
  • [11] G. F. Zhang, S. Zhang, B. F. Pan, X. F. Liu and L. S. Feng. Eur. J. Med. Chem. 2018, 143, 710.
  • [12] Y. X. Xu, H. Wang, X. K. Li, S. N. Dong, W. W. Liu, Q. Gong, T. D. Y. Wang, Y. Tang, J. Zhu, J. Li, H. Y. Zhang and F. Mao. Eur. J. Med. Chem. 2018, 143, 33.
  • [13] X. L. Hu, Z. Xu, M. L. Liu, L. S. Feng and G. D. Zhang. Curr. Top. Med. Chem. 2017, 17, 3219
  • [14] K. Wittine, M. S. Babić, D. Makuc, J. Plavec, S. K. Pavelić, M. Sedić, K. Pavelić, P. Leyssen, J. Neyts, J. Balzarini and M. Mintas. Bioorg. Med. Chem. 2012, 20, 3675
  • [15] E. Serrao, Z. L. Xu, B. Debnath, F. Christ, Z. Debyser, Y. Q. Long and N. Neamati. Bioorg. Med. Chem. 2013, 21, 5963
  • [16] J. Z. Vlahakis, R. T. Kinobe, K. Nakatsu, W. A. Szarek and I. E. Crandall. Bioorg. Med. Chem. Lett. 2016, 16, 2396
  • [17] Y. Q. Hu, C. Gao, S. Zhang, L. Xu, Z. Xu, L. S. Feng, X. Wu and F. Zhao. Eur. J. Med. Chem. 2017, 139, 22.
  • [18] A. Bistrović, L. Krstulović, A. Harej, P. Grbčić, M. Sedić, S. Koštrun, S. K. Pavelić, M. Bajić and S. Raić-Malić, Eur. J. Med. Chem. 2018, 143, 1616.
  • [19] R. Rajkumar, A.Kamaraj and K. Krishnasamy. Journal of Taibah University for Science, 2015, 9, 498.
  • [20] Vimalkumar H. Kapupara, Prakash L. Kalavadiya, Dinesh G. Gojiya, Nilesh D. Parmar, Hitendra S. Joshi. World Scientific News 119 (2019) 139-167

Document Type

article

Publication order reference

Identifiers

YADDA identifier

bwmeta1.element.psjd-e7fea9b8-fc69-44b0-9dc5-81f503527895
JavaScript is turned off in your web browser. Turn it on to take full advantage of this site, then refresh the page.