Synthesis of new derivatives of 9-(2-pyridyl)-3-aryl(arylalkyl)- -2,4,5(9H)trioxo-7,8-dihydroimidazo[1,2-a][1,3,5]triazepine

• Authors: Marzena Rzadkowska , Elzbieta Szacon , Maria Zun
• Languages of publication: EN

Abstracts

EN

A series of new derivatives of 9-(2-pyridyl)-3-aryl(arylalkyl)-2,4,5(9H)trioxo-7,8- dihydroimidazo [1,2-a][1,3,5] triazepine was obtained by condensation of 1-[1-(2-pyridyl) imidazolidine-2-ylidene]-3-aryl(arylalkyl)ureas) with diethyl oxalic acid ester. Considering the structure of the obtained compounds, it can be expected that these compounds can reveal pharmacological activity.

Keywords

EN

1-[1-(2-pyridyl)imidazolidine- 2-ylidene]-3-aryl(arylalkyl) ureas); derivatives; diethyl oxalic acid ester

• Publisher: De Gruyter Open
• Journal: Current Issues in Pharmacy and Medical Sciences
• Year: 2014
• Volume: 27
• Issue: 1
• Pages: 8-9

Dates

published

1 - 6 - 2014

received

16 - 1 - 2014

accepted

24 - 1 - 2014

online

30 - 5 - 2014

Contributors

author

Marzena Rzadkowska

• Chair and Department of Synthesis and Chemical Technology of Pharmaceutical Substances with Computer Modeling Unit, Faculty of Pharmacy with Division of Medical Analytics, Medical University of Lublin, Chodzki 4a, 20-093 Lublin, Poland

author

Elzbieta Szacon

• Chair and Department of Synthesis and Chemical Technology of Pharmaceutical Substances with Computer Modeling Unit, Faculty of Pharmacy with Division of Medical Analytics, Medical University of Lublin, Chodzki 4a, 20-093 Lublin, Poland

author

Maria Zun

• Chair and Department of Applied Pharmacy, Faculty of Pharmacy, Medical University of Lublin, Chodzki 1, 20-093 Lublin, Poland

References

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Identifiers

DOI

10.2478/cipms-2014-0002